Bringing Radiotracing to Titanium-Based Antineoplastics: Solid Phase Radiosynthesis, PET and ex Vivo Evaluation of Antitumor Agent [(45)Ti](salan)Ti(dipic)

Gregory Severin, Carsten H Nielsen, Andreas I Jensen, Jesper Fonslet, Andreas Kjær, Fedor Zhuravlev

39 Citationer (Scopus)

Abstract

We present a novel solid-phase based (45)Ti radiolabeling methodology and the implementation of (45)Ti-PET in titanium-based antineoplastics using the showcase compound [(45)Ti](salan)Ti(dipic). This development is intended to allow elucidation of the biodistribution and pharmacokinetics of promising new Ti-based therapeutics.

OriginalsprogEngelsk
TidsskriftJournal of Medicinal Chemistry
Vol/bind58
Udgave nummer18
Sider (fra-til)7591-5
Antal sider5
ISSN0022-2623
DOI
StatusUdgivet - 24 sep. 2015

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